Leuprolide acetate yog ib qho tshuaj agonist uas ua los ntawm cov tshuaj gonadotropin-releasing hormone (GnRH) uas ua haujlwm ntev thiab muaj kev sib raug zoo rau cov receptors pituitary GnRH. Nws txoj kev ua haujlwm yog nyob ntawm qhov ntau npaum li cas thiab lub sijhawm:
Kev piav qhia txog khoom
Leuprolide acetate yog ib qho tshuaj GnRH agonist uas ua raws li GMP, tsim tawm raws li cov qauv zoo nruj nrog cov ntaub ntawv DMF rau kev pom zoo los ntawm cov koom haum tswj hwm. Cov tshuaj peptide no (purity ≥98%) hloov kho cov tshuaj hormones, ntim ua hmoov dawb hauv cov fwj kaw. Khaws cia rau -20 ° C, nws zoo tagnrho rau kev tshawb fawb txog endocrinology thiab oncology. Siv rau R&D, xyuas kom ua raws li FDA cov lus qhia.
Cov cwj pwm
| Lub Npe Lus Askiv | Leuprolide acetate | Qhov Ceev | / |
| CAS TSIS MUAJ | 74381-53-6 | Cov Ntawv Qhia Txog Kev Hloov Pauv | / |
| Cov Qauv Molecular | C61H88N16O14 | Kev Khaws Cia | -20°C |
| Mol. wt. | 1269.47 | Kev yaj tau | MSO (Me ntsis), Methanol (Me ntsis) |
| EINECS No. | 686-285-8 | Daim Ntawv | Hmoov |
| MDL No. | MFCD00072080 | Xim | Dawb mus rau Off-White |
| Cov Ntsiab Lus Yaj | 150-155°C | Tus nqi PH | |
| Kev Ruaj Ntseg | Ruaj khov, tab sis huab cua rhiab heev thiab hygroscopic heev - khaws cia rau hauv qab argon. Tsis sib haum nrog cov kua qaub, acid chlorides, acid anhydrides, cov neeg sawv cev oxidizing. | ||
Txoj Haujlwm ntawm Kev Ua Haujlwm
Kev Txhawb Nqa Thaum Pib: Kev ua haujlwm luv luv ntawm cov pituitary GnRH receptors, ua rau muaj kev nce ntxiv ntawm luteinizing hormone (LH) thiab follicle-stimulating hormone (FSH) secretion.
Kev Tiv Thaiv Tom Qab: Kev siv ntev ntev ua rau cov receptors pituitary tsis ua haujlwm zoo, txo qis LH/FSH ntau lawm. Qhov no ua rau txo qis gonadal steroidogenesis (testosterone rau cov txiv neej, estrogen/progesterone rau cov poj niam), zoo li "kev txiav tawm hauv kev kho mob" rau lub hom phiaj kho mob.
Leuprolide acetate (GMP DMF) kho tau mob qog nqaij hlav prostate zoo los ntawm kev txo cov testosterone, ua rau cov qog loj hlob qeeb, thiab txo cov tsos mob xws li mob thiab tso zis tsis tau.
Nws pab tswj kev mob endometriosis los ntawm kev txwv tsis pub tsim cov tshuaj hormones hauv zes qe menyuam, txo qhov mob hauv plab thiab txo qhov loj ntawm qhov mob.
Hauv cov menyuam yaus, nws ncua kev loj hlob ntawm lub hnub nyoog laus hauv nruab nrab precious puberty, ua rau muaj kev loj hlob zoo dua.
Nws qhov zoo tau ntawv pov thawj GMP ua kom muaj kev nyab xeeb thiab ua haujlwm tau zoo hauv cov mob uas cuam tshuam nrog cov tshuaj hormones, txhawb nqa cov txiaj ntsig kho mob txhim khu kev qha.
Kev Loj Hlob Thaum Yau (CPP)
Kev Pab Txhawb Kev Tsim Me Nyuam (ART)

Txog Peb






Whatsapp
WeChat
